Custom Peptides
Cayman Chemical TrImetazIdInd8hydrochLRI 10mg
An internal standard for the quantification of trimetazidine by GC- or LC-MS
Cayman Chemical 2FluoroIsocathInonhydroch 10mg
A compound that structurally mimics substituted cathinones and phenethylamines; intended for research and forensic applications
Cayman Chemical 6-MAPBhydrochlorIde 10mg
An analytical reference standard categorized as a benzofuran; intended for research and forensic applications
Cayman Chemical Telbvudn 10mg
A β-L-nucleoside analog of thymidine that has antiviral activity; active against HBV in 2.2.15 cells (EC50 = 0.19 μM); selective for HBV over HIV-1, HSV-1, HSV-2, and influenza A and B (EC50s = >100 μM); reduces serum viral load in a woodchuck model of chronic HBV infection in a dose-dependent manner
Cayman Chemical GlucosdePNdent Insulnotro 10mg
A pro-atherogenic peptide; induces IκB-α degradation and NF-κB nuclear translocation in macrophage-differentiated THP-1 cells and isolated human aortic endothelial cells at 1 µM; increases atherosclerotic lesion area and plaque formation in ApoE-/- mice
Cayman Chemical notuberostemonIn 10mg
An alkaloid; inhibits LPS-induced increases in iNOS protein levels and NO production in RAW 264.7 cells at 100 µM; inhibits RANKL-induced osteoclast differentiation of RAW 264.7 cells at 50 µM; reduces the citric acid-induced cough reflex in conscious guinea pigs at 133 µmol/kg; inhibits pulmonary collagen deposition and fibrosis, as well as BALF monocyte and lymphocyte infiltration in a mouse model of bleomycin-induced pulmonary fibrosis at 40 mg/kg
Cayman Chemical McaKPLGLDap DnpARNH2tr 10mg
A fluorogenic substrate for MMPs; Mca is released upon cleavage by MMPs and its fluorescence can be used to quantify MMP activity; ex/em = 328/420 nm, respectively
Cayman Chemical 3 4dImethoxyaPyrroldInope 10mg
An analog of MDPV, differing only by an opening of the ring structure on the phenyl group; intended for research and forensic applications
Cayman Chemical 1 2DIoleoylsnglycero3PS 10mg
A phospholipid; SapC-1,2-DOPS nanovesicles are cytotoxic to SK-MEL-28 cells in vitro and decrease tumor volume in a squamous cell carcinoma mouse xenograft model; has been used in the formation of unilamellar vesicles to study the effect of curvature on membrane structure and in the formation of supported lipid bilayers to study the effects of various support materials on lipid redistribution between membrane leaflets
Cayman Chemical Pimpinellin 10mg
A coumarin derivative with diverse biological activities; inhibits AChE and BChE by 23.54 and 66.55%, respectively, at 20 UG/ml; inhibits collagen-induced aggregation of mouse platelets ex vivo at 40 mg/kg; inhibits PTZ-induced seizure-like behavior in zebrafish larvae
Cayman Chemical DaunorubIcInon 10mg
An aglcyone form of the antitumor antibiotic daunorubicin; has been used as a starting material in the synthesis of anticancer agents
Cayman Chemical PropylhexedrInhydrochLRId 10mg
An α-adrenergic sympathomimetic amine that acts as a local vasoconstrictor; intended for research and forensic applications
Cayman Chemical 9AmIno6chloro2methoxyacr 10mg
A fluorescent probe for DNA and pH gradients; selective for poly(dA-dT) sequences; has ex/em spectra of 411/475 nm, respectively; inhibits AChE (Ki = 49 nM)
Cayman Chemical BradykInInhumnmouserat 10mg
An endogenous vasodilator; binds to the bradykinin B2 receptor (IC50 = 0.54 nM in COS-7 cells expressing the human receptor) and acts as an agonist but does not bind the bradykinin B1 receptors (Ki = >10,000 nM in HEK293 cells expressing the human receptor); stimulates arachidonic acid release in CHO cells expressing the human bradykinin B2 receptor (EC50 = 0.7 nM); induces relaxation of ACh- or PDBu precontracted isolated porcine coronary arterial rings at 100 nM; induces hyperalgesia in mice at 1 UG/paw; plasma levels are increased in patients during an acute attack of angioedema
Cayman Chemical Enoctabn 10mg
A prodrug form of cytarabine; resistant to deamination by cytidine deaminase; reduces the virus yield in the supernatant of CMV-infected Vero cells (EC90 = 0.5 UG/ml); inhibits viral DNA synthesis at 5 UG/ml; increases survival in an L1210 murine skin lymphocytic leukemia model