Benzoxazines
TARGETMOL CHEMICALS INC INOBRODIB 5MG
Also available in 1 mg 2 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Inobrodib (CBP-IN-1) is a potent inhibitor of p300/CBP bromodomain. purity: 97%
TARGETMOL CHEMICALS INC DBPR112 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. DBPR112 is an orally active furanopyrimidine-based EGFR inhibitor with IC50s of 15 nM and 48 nM for EGFRWT and EGFRL858R/T790M respectively. DBPR112 can occupy the ATP-binding site. DBPR112 has significant antitumor efficacy. purity: 98%
TARGETMOL CHEMICALS INC FIVE1 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. FiVe1 is a vimentin binding small molecule that promotes the disintegration and phosphorylation of vimentin in the metaphase leading to mitotic disasters polynuclearization and loss of cancer cell dryness. FiVe1 selectively and irreversibly inhibit the growth of mesenchymal transformed breast cancer cells (FOXC2-HMLER cell IC50=234nM) and soft tissue sarcomas of different histological subtypes. purity: 98%
TARGETMOL CHEMICALS INC LUSUTROMBOPAG 5MG
Also available in 1 mg 2 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Lusutrombopag (Mulpleta) is an orally bioavailable small molecule thrombopoietin (TPO) receptor agonist for chronic liver disease (CLD) patients with thrombocytopenia prior to elective invasive surgery. purity: 99%
Medchemexpress LLC 7-Ethoxyresorufin | 5725-91-7 | 99.6% | 50 MG
7-Ethoxyresorufin, also known as Resorufin ethyl ether, is a fluorometric substrate and competitive inhibitor of cytochrome P450, specifically CYP1A1. It also inhibits NO synthase. This compound has been shown to reduce the relaxant actions of acetylcholine in endothelium-intact rings and of NO, GTN, and SNP in endothelium-denuded rings in rat aortic rings.
- Acts as a fluorometric substrate
- Functions as a competitive inhibitor of cytochrome P450, particularly CYP1A1
- Inhibits NO synthase
- Reduces the relaxant actions of acetylcholine, NO, GTN, and SNP
- Reacts with NADPH to produce a fluorescent product
TARGETMOL CHEMICALS INC ML-210 10MG
Also available in 1 mg 2 mg 5 mg 25 mg 50 mg 100 mg 200 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. ML-210 (CID 49766530) is a selective RAS and covalent glutathione peroxidase 4 (GPX4) inhibitor(GPX4 EC50 30 nM) with anti-cancer activitypurity: 97%
Medchemexpress LLC 7-Ethoxyresorufin | 5725-91-7 | 99.6% | 1 ML
7-Ethoxyresorufin is a fluorometric substrate and competitive inhibitor of cytochrome P450, especially CYP1A1. It also inhibits NO synthase. This compound is known for its role in biological activity and its fluorescent properties, making it suitable for various research applications.
- Fluorometric substrate
- Competitive inhibitor of cytochrome P450
- Inhibits NO synthase
- Reduces relaxant actions of acetylcholine
- Reacts with NADPH to form a fluorescent product
TARGETMOL CHEMICALS INC LESOPITRON 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Lesopitron is an anxiolytic with pre- and postsynaptic 5-HT1A agonist activity and is more effective than 5-HT1A agonists in rat social interaction and marmoset anxiety models. lesopitron counteracts benzodiazepine withdrawal-induced anxiety in rodents with low acute toxicity and does not potentiate the effects of alcohol or barbiturates. purity: 98%
TARGETMOL CHEMICALS INC THYMOPENTIN 10MG
Also available in 1 mg 2 mg 5 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Synthetic pentapeptide corresponding to the amino acids 32-36 of thymopoietin and exhibiting the full biological activity of the natural hormone. Thymopentin (TP5) is an immunomodulator which has been studied for possible use in the treatment of rheumatoid arthritis AIDS and other primary immunodeficiencies. purity: 99%
TARGETMOL CHEMICALS INC IQP-0528 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. IQP-0528 is a potent non-nucleoside reverse transcriptase inhibitor (NNRTI) that has potential for the treatment of HIV infection by blocking viral entry and shows antiviral activity as a microbicidal gel. . IQP-0528 showed inhibition of both HIV-1 and HIV-2 with an EC50 of 0.2 nM for HIV-1 and 100 nM for HIV-2. purity: 98%
TARGETMOL CHEMICALS INC ISORHAPONTIGENIN 10MG
Also available in 1 mg 5 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Isorhapontigenin (Isorhapotogenin) is a tetrahydroxylated stilbenoid with a methoxy group. It is an isomer of rhapontigenin and an analog of resveratrol. It is found in the Chinese herb Gnetum cleistostachyum in Gnetum parvifolium and in the seeds of the palm Aiphanes aculeata. purity: 99%