Cycloheptathiophenes
Medchemexpress LLC Formoterol fumarate | 43229-80-7 | >99.9% | C19H24N2O4 . 1/2C4H4O4 | 1 ML
Formoterol fumarate is a selective β2-adrenoceptor agonist, demonstrating similar β2-adrenoceptor selectivity to Salbutamol and Terbutaline. This compound is known for its ability to abolish the contraction induced by Acetylcholine in bronchioles. It is commonly utilized in research applications for conditions such as chronic obstructive pulmonary disease and bronchial asthma.
- Selective β2-adrenoceptor agonist
- Abolishes acetylcholine-induced contraction in bronchioles
- Used in research for chronic obstructive pulmonary disease
- Utilized in research for bronchial asthma
Medchemexpress LLC Tepilamide fumarate | 1208229-58-6 | 99.8% | 243.26 | 100 MG
Tepilamide fumarate is an oral fumaric acid ester that acts as a proagent of Monomethyl fumarate. It is used in the research of moderate to severe chronic plaque psoriasis and can enhance the effectiveness of oncolytic viruses.
- Oral fumaric acid ester
- Proagent of Monomethyl fumarate
- Enhances effectiveness of oncolytic viruses
- Selectively promotes oncolytic virus infection in cancer cells without affecting healthy tissues
- Used in research for moderate to severe chronic plaque psoriasis
- Potential to enhance virus-based therapy
- Solid, white to off-white appearance
Medchemexpress LLC Bedaquiline fumarate | 845533-86-0 | 99.99% | 671.58 | 1 ML
Bedaquiline fumarate, also known as R403323 or TMC207 fumarate, is a potent diarylquinoline antibiotic that primarily targets ATP synthase. This mechanism of action makes it highly effective for treating Mycobacterium tuberculosis infections, including difficult-to-treat multidrug-resistant (MDR) strains. It is intended for research use only.
- Antibiotic mechanism: Functions as a bacterial inhibitor by targeting ATP synthase
- Antituberculosis activity: Effective against Mycobacterium tuberculosis infections, including multidrug-resistant strains
- In vitro efficacy: Inhibits growth of TDR M. tuberculosis strains and shows high activity against Mycobacterium avium
- Research use: Intended for laboratory research and development
Apexbio Technology LLC Ro 60-0175 fumarate 169675-09-6 50mg
Ro 60-0175 fumarate (CAS 169675-09-6) is a selective agonist of the 5-HT2C serotonin receptor known to specifically activate serotonergic signaling pathways By targeting 5-HT2C receptors it modulates neurotransmitter release and neuronal circuitry influencing processes such as appetite regulation mood stabilization and cognitive function Ro 60-0175 fumarate is widely utilized in neuropharmacological research to investigate central nervous system mechanisms and to assess the pharmacological properties and therapeutic potential of 5-HT2C receptor agonists in models of depression anxiety obesity and related neuropsychiatric conditions
Medchemexpress LLC Bedaquiline fumarate | 845533-86-0 | 99.98% | 671.58 | 50 MG
Bedaquiline fumarate is an analytical standard and a diarylquinoline antibiotic that targets ATP synthase. It is effective for the treatment of Mycobacterium tuberculosis infections and is intended for research and analytical applications.
- Analytical standard grade
- Reference standard supplied assay
- Effective against Mycobacterium tuberculosis infections
- Commonly used in qualitative, quantitative, and methodological research experiments
- Suitable for HPLC, GC, and MS applications
Medchemexpress LLC Bedaquiline fumarate | 845533-86-0 | 99.99% | 671.58 | 5 MG
Bedaquiline fumarate is a diarylquinoline antibiotic that targets ATP synthase and is effective for the treatment of Mycobacterium tuberculosis infections.
- Inhibits the growth of TDR Mycobacterium tuberculosis strains.
- Highest activity against Mycobacterium avium among slowly growing mycobacteria.
- Shows moderate in vitro activity against NTM species.
- Excellent in vitro activity against multidrug-resistant Mycobacterium tuberculosis.
Medchemexpress LLC Diethyl fumarate | 623-91-6 | 99.0% | 172.18 | 10 G
Diethyl fumarate is a decomposition product of Malathion 9 and a reactant in the Diels-Alder reaction. It is a reputed skin irritant and can cause non-immunologic contact urticaria on the skin. Diethyl fumarate and Curcumin hybridize to exert neuroprotective effects.
- Decomposition product of Malathion 9.
- Reactant in Diels-Alder reaction.
- Causes dose-dependent swelling of ears in guinea pigs.
- Curcumin hybrids show neuroprotective effects in C. elegans model of PD.
- For research use only.
Medchemexpress LLC Cevipabulin fumarate | 849550-67-0 | 99.9% | 580.89 | 50 MG
Cevipabulin fumarate (TTI-237 fumarate) is an oral, microtubule-active, antitumor compound. It inhibits the binding of [3H]NSC 49842 to tubulin, with an IC50 of 18-40 nM for cytotoxicity in human tumor cell lines.
- Microtubule-active, antitumor compound
- Shows good activity (18-40 nM IC50 values) on ovarian, breast, prostate, and cervical tumor cell lines
- Produces sub-G1 nuclei at low concentrations (20-40 nM)
- Causes a strong G2-M block at concentrations above 50 nM
- Active via intravenous (i.v.) and oral (p.o.) administration against human tumor xenografts in mice, with good antitumor activity at 20 and 15 mg/kg
Medchemexpress LLC Iron(II) fumarate (Ferrous fumarate) | 141-01-5 | 95.1% | 1 G
Iron (II) fumarate is an orally effective active dietary supplement. It can alleviate metabolic damage and damage to silkworms caused by cypermethrin and can be used for research on iron deficiency anemia.
- In vitro: Can restore metabolic pathway disruption and enhance cell viability in BmN cells treated with cypermethrin.
- In vivo: Alleviates damage caused by cypermethrin in silkworms.
- In vivo: Induces oxidative stress in the liver and colon of rats.
- In vivo: Alters intestinal morphology and microbiota in Yellow River carp, increasing diversity and richness.
Medchemexpress LLC Formoterol fumarate | 43229-80-7 | >99.9% | C19H24N2O4 . 1/2C4H4O4 | 100 MG
Formoterol fumarate is a selective β2-adrenoceptor agonist, at least as selective as Salbutamol and Terbutaline. It relaxes acetylcholine-pre-contracted human isolated segmental bronchi and can be used for research related to chronic obstructive pulmonary disease and bronchial asthma.
- Selective β2-adrenoceptor agonist
- Relaxes acetylcholine-pre-contracted human isolated segmental bronchi
- Suitable for research on chronic obstructive pulmonary disease
- Suitable for research on bronchial asthma
Medchemexpress LLC Diroximel fumarate | 1577222-14-0 | ≥98.0% | 255.23 g/mol | C11H13NO6 | 50 MG
Diroximel fumarate is supplied as a research-grade small-molecule reagent intended for laboratory studies. This listing represents a 50 MG pack of the prodrug of monomethyl fumarate and is provided for experimental and analytical use in research settings; it is not for clinical or human use.
- For research use only, not for human or clinical use.
- Supplied as a small 50 MG pack suitable for laboratory testing.
- High purity, typically ≥98.0%.
- Molecular weight 255.23 g/mol and formula C11H13NO6.
- Useful for studies of fumarate metabolism and related biochemical pathways.
Medchemexpress LLC Formoterol fumarate | 43229-80-7 | 99.8% | C19H24N2O4·1/2C4H4O4 | 50 MG
Formoterol fumarate is a selective β2-adrenoceptor agonist. This compound abolishes contraction induced by Acetylcholine in bronchioles and can be utilized for research into chronic obstructive pulmonary disease and bronchial asthma.
- Selective β2-adrenoceptor agonist
- Abolishes contraction induced by Acetylcholine in bronchioles
- Can be used for research of chronic obstructive pulmonary disease and bronchial asthma
- Appears as a white to off-white solid
- Soluble in DMSO at ≥ 50 mg/mL
Apexbio Technology LLC Ibutilide Fumarate 122647-32-9 100mg
Ibutilide Fumarate (CAS 122647-32-9) is a small molecule classified as a Class III antiarrhythmic agent It acts primarily by enhancing slow inward sodium currents and delaying repolarization through inhibition of the rapid component of the cardiac delayed rectifier potassium current (IKr) resulting in prolongation of the cardiac action potential Ibutilide is utilized in research to investigate pharmacological cardioversion of atrial arrhythmias specifically studying the acute conversion of atrial fibrillation and atrial flutter to normal sinus rhythm Its properties make it valuable for exploring the mechanisms of antiarrhythmic therapy and cardiac electrophysiology
Selleck Chemical LLC Ketotifen Fumarate S2024-50mg
Ketotifen Fumarate(HC 20511 fumarate) is a fumaric acid salt of ketotifen which is a H1-antihistamine and mast cell stabilizer