Piperidines
eMolecules 19365-08-3 | 3-Hydroxy-2-piperidinone | AA Blocks LLC | MFCD00023163 | 115.132 | C5H9NO2 | 0.000 | OC1CCCNC1=O | 250mg | 425799725
3-Hydroxy-2-piperidinone | AA Blocks LLC | 19365-08-3 | MFCD00023163 | 115.132 | C5H9NO2 | 0.000 | OC1CCCNC1=O | 250mg | 425799725
Medchemexpress LLC Piperidin-2-one | 675-20-7 | 99.9% | 99.13 g/mol | C5H9NO | 10 G
2-Piperidone (piperidin-2-one; δ-valerolactam) is an endogenous metabolite and a biomarker for CYP2E1 activity. It is supplied as a high-purity research standard for use in analytical, metabolic, and pharmacological studies. CAS number 675-20-7; molecular formula C5H9NO; molecular weight 99.13 g/mol; purity 99.89%.
- high-purity research-grade material suitable for analytical assays and reference standards.
- soluble in DMSO and water at high concentrations with ultrasonic aid.
- provided in multiple pack sizes to support small-scale and bulk experiments.
- storage recommendations available for long-term stability in solid and solvent forms.
Accela Chembio Inc N-boc-4-nortropinone | 25g | 185099-67-6 | MFCD00673779 | 98% | Shelf Life: 1980 Days | Regular
N-boc-4-nortropinone | 25g | 185099-67-6 | MFCD00673779 | 98% | Shelf Life: 1980 Days | Regular
Medchemexpress LLC Bsj-03-204 | 2349356-09-6 | 99.76% | 832.90 | 100 MG
BSJ-03-204 is a PROTAC (proteolysis-targeting chimera) that connects ligands for Cereblon and CDK. It is a potent and selective Palbociclib-based CDK4/6 dual degrader, demonstrating anti-cancer activity and potent anti-proliferative effects on MCL cell lines.
- Potent and selective Palbociclib-based CDK4/6 dual degrader
- Does not induce IKZF1/3 degradation
- Exhibits anti-cancer activity
- Potent anti-proliferative effects on MCL cell lines
- Induces a G1 arrest
Medchemexpress LLC 2-piperidone | 675-20-7 | MFCD00006037 | 99.9% | 99.13 g/mol | C5H9NO | 25 G
2-Piperidone is a small lactam (δ-valerolactam) used as a research reagent and a biomarker for CYP2E1 activity. It is provided as a high-purity reference standard suitable for in vitro and in vivo metabolic studies and formulation development.
- CAS number 675-20-7.
- Purity 99.9%.
- Molecular formula C5H9NO.
- Molecular weight 99.13 g/mol.
- Solubility: DMSO and water 100 mg/mL (ultrasonic recommended); in vivo formulations ≥2.5 mg/mL in common vehicles.
- Storage: pure form -20°C (3 years), 4°C (2 years); in solvent -80°C (6 months), -20°C (1 month).
- Available pack sizes include 25 g.
Medchemexpress LLC TD-0212 TFA 10mg | 1073549-11-7 | 10 MG
TD-0212 TFA is a research-grade small molecule supplied as the trifluoroacetate (TFA) salt that acts as an orally active dual angiotensin II type 1 (AT1) receptor antagonist and neprilysin (NEP) inhibitor. It is provided as a white to off-white solid for laboratory research use only.
- Dual AT1 antagonist and NEP inhibitor with reported pKi 8.9 and pIC50 9.2.
- High purity (98.44%) suitable for biological research.
- Molecular formula C30H35F4N3O6S; molecular weight 641.67.
- Soluble in DMSO (125 mg/mL) and compatible with in vivo co-solvent preparation protocols.
- Stable when stored sealed at -20°C; in solution store at -80°C for long term.
Enzo Life Sciences dBET1 (100mg). CAS: 1799711-21-9
dBET1 is a PROTAC, consisting of a BRD4-ligand JQ-1 linked to a cereblon E3 ligase ligand, targeting on BET bromodomain BRD4. Purity: ≥99%. Long Term Storage: -20°C.
Medchemexpress LLC BSJ-4-116 | 2519823-34-6 | 99.9% | 837.38 | 100 MG
BSJ-4-116 | 2519823-34-6 | 99.9% | 837.38 | 100 MG
Medchemexpress LLC Gemigliptin tartrate | 1374639-74-3 | 99.5% | 639.45 | 50 MG
Gemigliptin tartrate is a highly selective, reversible, and competitive dipeptidyl peptidase-4 (DPP-4) inhibitor with an IC50 of 10.3 nM for human recombinant DPP-4. It exhibits potent anti-glycation properties and can be utilized for research into advanced glycation end products (AGE)-related diabetic complications.
- Highly selective, reversible, and competitive DPP-4 inhibitor
- Exhibits potent anti-glycation properties
- Can be used for research into advanced glycation end products (AGE)-related diabetic complications
- Inhibits the formation of AGE-BSA
- Suppresses the cross-linking of preformed AGE-BSA
- Dose-dependently inhibits plasma DPP-4 activity in rats, dogs, and monkeys
- Significantly reduces circulating AGE levels in serum in vivo
Medchemexpress LLC Pomalidomide-C12-NH2 hydrochloride | 2862774-02-3 | 97.1% | 493.04 g/mol | C25H37ClN4O4 | 5 MG
Pomalidomide-C12-NH2 hydrochloride is an E3 ligase ligand-linker conjugate used as the Cereblon-directed ligand component in PROTAC design targeting KRAS G12C. Supplied as the hydrochloride salt for research use, it is provided as a solid in milligram scales and is characterized by high purity and defined storage recommendations.
Medchemexpress LLC HY-50667 1g , Apixaban BMS-562247-01 CAS:503612-47-3 Purity:98%
Medchemexpress, HY-50667 1g Apixaban BMS-562247-01 CAS:503612-47-3 Formula:C25H25N5O4 IC50: 0.08 nM (Human Factor Xa), 0.17 nM (Rabbit Factor Xa) Purity:98% Apixaban is a highly selective, reversible inhibitor of Factor Xa with K i of 0.08 nM and 0.17 nM in human and rabbit, respectively. Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC 2-piperidinone | 675-20-7 | MFCD00006037 | ≥98.0% | 99.13 g/mol | C5H9NO | 500 G
2-piperidinone is an endogenous metabolite and a biomarker for CYP2E1 activity, supplied as a research-grade solid with high purity and DMSO solubility.
- Endogenous metabolite and CYP2E1 biomarker.
- Solid powder suitable for laboratory use.
- Purity ≥98.0% (reported by manufacturer).
- Molecular weight 99.13 g/mol and formula C5H9NO.
- Soluble in DMSO at approximately 100 mg/mL; may require ultrasonic assistance.
- Store powder at -20°C for long-term stability; in solution keep at -80°C.
Medchemexpress LLC FGI-106 tetrahydrochloride | 1149348-10-6 | 99.7% | 604.49 g/mol | C28H42Cl4N6 | 5MG
FGI-106 tetrahydrochloride is a research-grade, broad-spectrum antiviral inhibitor supplied as the tetrahydrochloride salt for in vitro studies. It has reported activity against several viral pathogens and is intended for laboratory research use only. Prepare stocks in DMSO following solubility guidance and handle per standard laboratory safety procedures.
- Cas number 1149348-10-6.
- Molecular formula C28H42Cl4N6; molecular weight 604.49 g/mol.
- Purity approximately 99.7%.
- Appearance solid, light brown to brown.
- Soluble in DMSO with heating, ultrasonication, and pH adjustment; reported solubility 6.67 mg/mL in DMSO.
- Recommended stock concentrations: 1 mM, 5 mM, and 10 mM in DMSO with mg-to-mL conversion guidance.
- Store sealed, away from moisture; in solvent: -80°C up to 6 months, -20°C up to 1 month.
- For research use only; not for human or clinical use.