Bioactive Small Molecules
Medchemexpress LLC HY-50514 2mg , AT9283 CAS:896466-04-9 Purity:>98%
HY-50514 2mg AT9283 CAS: 896466-04-9 AT9283 is a multi-targeted kinase inhibitor with potent activity against Aurora A/B, JAK2/3, Abl (T315I) and Flt3 (IC50s ranging from 1 to 30 nM). AT9283 inhibits growth and survival of multiple solid tumors in vitro and in vivo. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-112726 5mg , PXS-4728A CAS:1478364-68-9 Purity:>98%
HY-112726 5mg PXS-4728A CAS: 1478364-68-9 PXS-4728A (BI-1467335) is a selective, orally active inhibitor of semicarbazide-sensitive amine oxidase (SSAO). PXS-4728A ameliorates chronic obstructive pulmonary disease in mice. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-116770 10mg , PFM01 CAS:1558598-41-6 Purity:>98%
HY-116770 10mg PFM01 CAS: 1558598-41-6 PFM01, N-alkylated Mirin derivative, is a MRE11 endonuclease inhibitor. PFM01 can regulate double-strand break repair (DSBR) by nonhomologous end-joining (NHEJ) versus homologous recombination (HR). Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-P0210 5mg , DAMGO CAS:78123-71-4 Purity:>98%
HY-P0210 5mg DAMGO CAS: 78123-71-4 DAMGO is a μ-opioid receptor (μ-OPR ) selective agonist with a Kd of 3.46 nM for native μ-OPR. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-132001 5mg , Ziftomenib CAS:2134675-36-6 Purity:>98%
HY-132001 5mg Ziftomenib CAS: 2134675-36-6 Ziftomenib (KO-539) is a menin-MLL interaction inhibitor with antitumor activities (WO2017161028A1, compound 151). Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-15465 1mg , KN-93 CAS:139298-40-1 Purity:>98%
HY-15465 1mg KN-93 CAS: 139298-40-1 KN-93 is a cell-permeable, reversible and competitive inhibitor calmodulin-dependent kinase type II (CaMKII) with a Ki of 370 nM. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-70002 5g , Enzalutamide CAS:915087-33-1 Purity:>98%
HY-70002 5g Enzalutamide CAS: 915087-33-1 Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells. Enzalutamide is an autophagy activator. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-13901 10mg , GANT 61 CAS:500579-04-4 Purity:>98%
HY-13901 10mg GANT 61 CAS: 500579-04-4 GANT 61 is an inhibitor of Gli1 and Gli2 targeting the Hedgehog/GLI pathway. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-139399 5mg , JNJ-67856633 CAS:2230273-76-2 Purity:>98%
HY-139399 5mg JNJ-67856633 CAS: 2230273-76-2 JNJ-67856633 is an orally active, first-in-class, potent, selective and allosteric MALT1 protease inhibitor. JNJ-67856633 in some cases lead to tumor stasis. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-13319 2mg , JNK-IN-8 CAS:1410880-22-6 Purity:>98%
HY-13319 2mg JNK-IN-8 CAS: 1410880-22-6 JNK-IN-8 (JNK Inhibitor XVI) is a potent JNK inhibitor with IC50s of 4.7 nM, 18.7 nM, and 1 nM for JNK1, JNK2, and JNK3, respectively. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-103683 10mg , PF-06409577 CAS:1467057-23-3 Purity:>98%
HY-103683 10mg PF-06409577 CAS: 1467057-23-3 PF-06409577 is a potent and selective allosteric activator of AMPK α1β1γ1 isoform with an EC50 of 7 nM. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-139567 5mg , Afimetoran CAS:2171019-55-7 Purity:>98%
HY-139567 5mg Afimetoran CAS: 2171019-55-7 Afimetoran is a toll-like receptor antagonist, which can be used in the research of inflammatory and autoimmune diseases. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-15605 1mg , Encorafenib CAS:1269440-17-6 Purity:>98%
HY-15605 1mg Encorafenib CAS: 1269440-17-6 Encorafenib (LGX818) is a highly potent BRAF inhibitor with selective anti-proliferative and apoptotic activity in cells expressing BRAFV600E (EC50=4 nM). Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-15659 10mg , Wnt-C59 CAS:1243243-89-1 Purity:>98%
HY-15659 10mg Wnt-C59 CAS: 1243243-89-1 Wnt-C59 (C59) is a highly potent and oral porcupine (PORCN) inhibitor with an IC50 of 74 pM. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-15741 1mg , Mc-MMAE CAS:863971-24-8 Purity:>98%
HY-15741 1mg Mc-MMAE CAS: 863971-24-8 Mc-MMAE is a protective group (maleimidocaproyl)-conjugated monomethyl auristatin E (MMAE), which is a potent tubulin inhibitor. Mc-MMAE is a drug-linker conjugate for ADC. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.