Bioactive Small Molecules

A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.

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6,706 – 6,720 of 60,541 results

6,706

AdipoGen Kendomycin

Chemical. CAS 183202-73-5. Formula C29H42O6. MW 486.6. Isolated from Streptomyces violaceoruber. Antibiotic. Potent endothelin receptor antagonist. Anti-osteoporotic. Antibacterial. Cytotoxic. Mediates its cytotoxic effects, at least in part, through proteasome inhibition.

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6,707

AdipoGen Telithromycin

Chemical. CAS 191114-48-4. Formula C43H65N5O10. MW 812. Semi-synthetic. Ketolide type macrolide antibiotic. Antibacterial compound used to treat mild to moderate respiratory infections. Protein synthesis inhibitor, by binding to the 50S ribosomal subunit and subsequently blocking the progression of the growing polypeptide chain. Binds to domains II and V of the 23S rRNA of the 50S ribosomal subunit. Has a higher affinity for these ribosomal targets than conventional macrolides due to the additional interactions and increased binding at domain II. Retains activity against Gram-positive cocci in the presence of resistance mediated by methylases erm genes that alter the binding site at domain V. May inhibit the formation of ribosomal subunits 50S and 30S.

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6,708

AdipoGen IronIII ionophore VI

Chemical. CAS 938155-11-4. Formula C23H20N2O. MW 340.4. Synthetic. Iron III ionophore dye.

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6,709

AdipoGen AMCA-X

Chemical. CAS 205124-69-2. Formula C18H22N2O5. MW 346.38. Synthetic. Amine-reactive blue fluorescent probe.

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6,710

AdipoGen Luteoreticulin

Chemical. CAS 22388-89-2. Formula C19H19NO5. MW 341.4. Isolated from Streptomyces thioluteus. Nitrophenyl pyranone derivative related to aureothin Prod. No. BVT-0303 http//www.adipogen.com/bvt-0303/aureothin.html . Insecticidal and nematocidal compound. Metabolites within this product class show pronounced antitumor and immunosuppressive activity.

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6,711

Medchemexpress LLC Samuraciclib hydrochloride hydrate | 00-00-0 | 99.9% | 552.33 | C22H33ClN6O2 | 5 MG

Samuraciclib hydrochloride hydrate is the hydrochloride hydrate salt of samuraciclib, a potent, selective, ATP-competitive, orally active CDK7 inhibitor used for research. It inhibits CDK7 with an IC50 of 41 nM, shows selectivity versus related cyclin-dependent kinases, and reduces proliferation of breast cancer cell lines (GI50 0.2-0.3 μM).

Potent CDK7 inhibition (IC50 41 nM).
Selective versus CDK1, CDK2, CDK5, and CDK9.
Demonstrated cellular activity in breast cancer cell lines (GI50 0.2-0.3 μM).
High chemical purity (99.88%).
Hydrochloride hydrate salt form for improved handling.
Available in small research pack sizes suitable for in vitro studies.

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6,712

Medchemexpress LLC L-Hydroxyproline (Standard) | 51-35-4 | 99.9% | 131.13 | 50 MG

L-Hydroxyproline (Standard) is the analytical standard of L-Hydroxyproline. This product is intended for research and analytical applications. L-Hydroxyproline, one of the hydroxyproline (Hyp) isomers, is a useful chiral building block in the production of many pharmaceuticals.

The compound is the grade of analytical standard, which is the reference standard supplied assay. It is commonly used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS.
Structure classification: Alkaloids, Pyrrole Alkaloids.
Initial source: Endogenous metabolite, Disease markers, Endocrine diseases, Nervous System Disorder, Immune System Disorder.

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6,713

Medchemexpress LLC YAP/TAZ inhibitor-3 | 2506273-81-8 | 99.3% | 389.37 | 10 MM X 1 ML

YAP/TAZ inhibitor-3 | 2506273-81-8 | 99.3% | 389.37 | 10 MM X 1 ML

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6,714

Medchemexpress LLC Indole-3-carboxylic acid | 771-50-6 | 99.6% | 161.16 | 5 MG

Indole-3-carboxylic acid (Standard) is the analytical standard of Indole-3-carboxylic acid. It is intended for research and analytical applications. Indole-3-carboxylic acid is a normal urinary indolic tryptophan metabolite and has been found to be elevated in patients with liver diseases. The compound is of analytical standard grade, used as a reference in qualitative, quantitative, and methodological research experiments, particularly in HPLC, GC, and MS.

Analytical standard for Indole-3-carboxylic acid.
Intended for research and analytical applications.
Used in qualitative, quantitative, and methodological research experiments (HPLC, GC, MS).

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6,715

Medchemexpress LLC Metaxalone | 1665-48-1 | 99.8% | 50 MG

Metaxalone is an FDA-approved muscle relaxant that primarily acts on the central nervous system by inhibiting polysynaptic reflex arcs. It also functions as an inhibitor of MAO-A, demonstrating anti-inflammatory and antioxidant effects. This product is for research use only.

Inhibits polysynaptic reflex arcs
Acts as an inhibitor of MAO-A
Demonstrates anti-inflammatory and antioxidant effects
Inhibits IL-1β-induced inflammatory phenotype
Modulates NF-κB and other related signaling pathways
Decreases MAO-A expression and activity in IL-1β-treated microglia

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6,716

Medchemexpress LLC Barium sulfate | 7727-43-7 | 99.0% | 500 G

Barium sulfate (Baryta white) is a biological material or organic compound that can be used as an opacifier. It is widely used in life science research.

Can be used as an opacifier
Widely used in life science research

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6,717

Medchemexpress LLC Deferiprone | 30652-11-0 | 100.0% | 100 MG

Deferiprone | 30652-11-0 | 100.0% | 100 MG

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6,718

Selleck Chemical LLC BMS-986278-E1036-5MG

BMS-986278 is a potent and orally active antagonist of lysophosphatidic acid receptor 1 (LPA1) BMS-986278 exhibits Kbs of 6 9 nM and 4 0 nM for human and mouse LPA1 respectively and is widely used in the research of pulmonary fibrotic diseases

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6,719

Selleck Chemical LLC Sotorasib (AMG510) 25mg 2296729-00-3

Sotorasib (AMG510) is a potent KRAS G12C covalent inhibitor with potential antineoplastic activity.This AMG510 is a chiral compound. *For Research & Development use only. Product is not intended for drug, household, or human consumption.

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6,720

Invivogen 2'3'-cGAMP, Mammalian (non-canonical) CDN, cyclic [G(2’,5’)pA(3’,5’)p], 1441190-66-4, MFCD31563596, 200 µg

Formula: C20H22N10O13P2 .2Na, Purity: ≥ 95% by LC/MS, Molecular weight: 718.38, 2’3’-cGAMP (cyclic [G(2’,5’)pA(3’,5’)p]) is produced in mammalian cells by cGAS (cGAMP synthase) in response to double-stranded DNA in the cytoplasm. It is also referred to as “noncanonical“ cGAMP due to the presence of the atypical 2’-5’ phosphodiester linkage between the guanosine and the adenosine.

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Bioactive Small Molecules

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Medchemexpress LLC Samuraciclib hydrochloride hydrate | 00-00-0 | 99.9% | 552.33 | C22H33ClN6O2 | 5 MG Small and Specialty Supplier PartnerSmall and/or specialty supplier based on Federal laws and SBA requirements.Learn More

Medchemexpress LLC L-Hydroxyproline (Standard) | 51-35-4 | 99.9% | 131.13 | 50 MG Small and Specialty Supplier PartnerSmall and/or specialty supplier based on Federal laws and SBA requirements.Learn More

Medchemexpress LLC YAP/TAZ inhibitor-3 | 2506273-81-8 | 99.3% | 389.37 | 10 MM X 1 ML Small and Specialty Supplier PartnerSmall and/or specialty supplier based on Federal laws and SBA requirements.Learn More

Medchemexpress LLC Indole-3-carboxylic acid | 771-50-6 | 99.6% | 161.16 | 5 MG Small and Specialty Supplier PartnerSmall and/or specialty supplier based on Federal laws and SBA requirements.Learn More

Medchemexpress LLC Metaxalone | 1665-48-1 | 99.8% | 50 MG Small and Specialty Supplier PartnerSmall and/or specialty supplier based on Federal laws and SBA requirements.Learn More

Medchemexpress LLC Barium sulfate | 7727-43-7 | 99.0% | 500 G Small and Specialty Supplier PartnerSmall and/or specialty supplier based on Federal laws and SBA requirements.Learn More

Medchemexpress LLC Deferiprone | 30652-11-0 | 100.0% | 100 MG Small and Specialty Supplier PartnerSmall and/or specialty supplier based on Federal laws and SBA requirements.Learn More