Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,276
Tocris Bioscience™ ST 045849
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O-GlcNAc transferase (OGT) inhibitor
| CAS | 442665-87-4 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 2-[(4-Chlorophenyl)imino]tetrahydro-4-oxo-3-(2-tricyclo[3.3.1.13,7]dec-1-ylethyl)-2H-1,3-thiazine-6-carboxylic acid |
| Molecular Formula | C23H27ClN2O3S |
1,277
Tocris Bioscience™ ML 252
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective KV7.2 inhibitor; brain penetrant
| Target | Voltage-gated Potassium Channel Blockers |
|---|---|
| CAS | 1392494-64-2 |
| Purity | 0.98 |
| Chemical Name or Material | (S)-2-Phenyl-N-(2-(pyrrolidin-1-yl)phenyl)butanamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C20H24N2O |
1,278
Tocris Bioscience™ SIS3
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Selective Smad3 inhibitor; inhibits TGF-βR1 signaling
| Product Type | SIS3 |
|---|---|
| Molecular Weight (g/mol) | 489.99 |
| Purity | 97% |
1,279
Tocris Bioscience™ 4μ8C
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CAS: 14003-96-4 Molecular Formula: C11H8O4
| CAS | 14003-96-4 |
|---|---|
| Molecular Formula | C11H8O4 |
1,280
Tocris Bioscience™ Ro 48-8071 fumarate
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2,3-Oxidosqualene cyclase (OSC) inhibitor; blocks cholesterol synthesis
| Inhibitors | Ro 48-8071 fumarate |
|---|---|
| CAS | 189197-69-1 |
| Product Type | Ro 48-8071 fumarate |
| Molecular Weight (g/mol) | M.W. (Observed): 564.44 |
| Purity | 99% |
| Recommended Storage | 4°C |
| Molecular Formula | (4-Bromophenyl)[2-fluoro-4-[[6-(methyl-2-propen-1-ylamino)hexyl]oxy]phenyl]methanone |
1,281
Tocris Bioscience™ Thalidomide 4'-ether-PEG2-azide
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Cereblon ligand with PEG linker and terminal azide for onward chemistry
1,282
Tocris Bioscience™ FURA-2AM
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CAS: 108964-32-5 Molecular Formula: C44H47N3O24
| CAS | 108964-32-5 |
|---|---|
| Molecular Formula | C44H47N3O24 |
1,283
Tocris Bioscience™ PD 173074
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 219580-11-7 Molecular Formula: C28H41N7O3
| CAS | 219580-11-7 |
|---|---|
| Molecular Formula | C28H41N7O3 |
1,284
Tocris Bioscience™ NK 252
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Nrf2 activator
| CAS | 1414963-82-8 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in 1eq. HCl and to 100mM in DMSO |
| Purity | >98% |
| Physical Form | Powder |
| Chemical Name or Material | NK 252 |
| Recommended Storage | Store at 4°C |
| Synonym | N-[5-(2-Furanyl)-1,3,4-oxadiazol-2-yl]-N'-(2-pyridinylmethyl)urea |
| Molecular Formula | C13H11N5O3 |
| Formula Weight | 285.26 |
1,285
Tocris Bioscience™ PR 619
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Broad spectrum DUB inhibitor
| CAS | 2645-32-1 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 10mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | PR 619 |
| Recommended Storage | Store at -20°C |
| Synonym | 2,6-Diamino-3,5-dithiocyanopyridine |
| Molecular Formula | C7H5N5S2 |
| Formula Weight | 223.28 |
1,286
Tocris Bioscience™ Phentolamine Mesylate
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Adrenergic α receptor antagonist; antihypertensive
1,287
Tocris Bioscience™ ML 9 hydrochloride
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CAS: 105637-50-1 Molecular Formula: C15H18Cl2N2O2S
| CAS | 105637-50-1 |
|---|---|
| Molecular Formula | C15H18Cl2N2O2S |
1,288
Tocris Bioscience™ Chromanol 293B
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CAS: 163163-23-3 Molecular Formula: C15H20N2O4S
| CAS | 163163-23-3 |
|---|---|
| Molecular Formula | C15H20N2O4S |
1,289
Tocris Bioscience™ E-4031 dihydrochloride
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CAS: 113559-13-0 Molecular Formula: C21H29Cl2N3O3S
| CAS | 113559-13-0 |
|---|---|
| Molecular Formula | C21H29Cl2N3O3S |
1,290
Tocris Bioscience™ A 804598
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CAS: 1125758-85-1 Molecular Formula: C19H17N5
| CAS | 1125758-85-1 |
|---|---|
| Molecular Formula | C19H17N5 |