Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Ezh2/Ezh1 Inhibitor, UNC1999
A cell-permeable GSK126 structural analog
MilliporeSigma™ Calbiochem™ PD 158780
A potent, cell-permeable, reversible, ATP-competitive inhibitor of the EGFR tyrosine kinase activity (IC50 = 8 pM).
MilliporeSigma™ Calbiochem™ Protease Inhibitor Cocktail Set V, Animal-Free
The Protease Inhibitor Cocktail Set V, Animal-Free controls the activity of Protease. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ MG-115
Potent reversible proteasome inhibitor (Ki = 21 nM and 35 nM for 20S and 26S proteasome, respectively).
MilliporeSigma™ Calbiochem™ GPR40 Antagonist, GW1100
The GPR40 Antagonist, GW1100, also referenced under CAS 306974-70-9, controls the biological activity of GPR40. This small molecule/inhibitor is primarily used for Biochemicals applications.
MilliporeSigma™ Calbiochem™ Chymotrypsin Substrate II, Fluorogenic
Sensitive fluorogenic substrate for the quantitative determination of chymotrypsin activity.
MilliporeSigma™ Calbiochem™ MPS1 Inhibitor III, AZ3146
A cell permeable purinone derivative that acts as a highly potent and selective inhibitor of monopolar spindle 1 kinase (MPS1; IC50 = ∽35
MilliporeSigma™ Calbiochem™ Cdc25 Inhibitor IV, NSC 95397
The Cdc25 Inhibitor IV, NSC 95397, also referenced under CAS 93718-83-3, controls the biological activity of Cdc25. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ TTNPB
A synthetic stilbene analog of retinoic acid that acts as a potent retinoic acid receptor (RAR) agonist (EC50 = 21 nM, 4.0 nM, and 2.4nM for RARα, RARβ, and RARγ, respectively).
MilliporeSigma™ Calbiochem™ DNA Base Excision Repair Pathway Inhibitor
The DNA Base Excision Repair Pathway Inhibitor, also referenced under CAS 6960-45-8, controls the biological activity of APE1 (human apurinic/apyrimidinic endonuclease.
MilliporeSigma™ Calbiochem™ Tankyrase1/2 Inhibitor IV, JW55
The Tankyrase1/2 Inhibitor IV, JW55 controls the biological activity of Tankyrase1/2. This small molecule/inhibitor is primarily used for Biochemicals applications.
MilliporeSigma™ Calbiochem™ GM 6001, Negative Control
A useful negative control for the MMP inhibitor GM 6001.
MilliporeSigma™ Calbiochem™ QX-314
A quaternary lidocaine derivative, permanently charged, and lipophobic.
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MilliporeSigma™ Calbiochem™ α2-Macroglobulin, Human Plasma
A multifunctional, secreted glycoprotein that acts as a broad range irreversible protease inhibitor that forms a trap around most proteases.
MilliporeSigma™ Calbiochem™ Aurora Kinase/Cdk Inhibitor
The Aurora Kinase/Cdk Inhibitor, also referenced under CAS 443797-96-4, controls the biological activity of Aurora Kinase/Cdk. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.