Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ HDL Receptor SR-BI Inhibitor, BLT-1
The HDL Receptor SR-BI Inhibitor, BLT-1, also referenced under CAS 321673-30-7, controls the biological activity of HDL Receptor SR-B. This small molecule/inhibitor is primarily used for Phosphorylation and Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Kaempferol
A cell-permeable phytoestrogen that inhibits topoisomerase I-catalyzed DNA religation in HL-60 cells.
MilliporeSigma™ Calbiochem™ TrkB Agonist, 7,8-Dihydroxyflavone
A cell permeable flavone based compound with neurotrophic and neuroprotective properties
MilliporeSigma™ Calbiochem™ eIF-2α Inhibitor II, Sal003
The eIF-2α Inhibitor II, Sal003, also referenced under CAS 301359-91-1, controls the biological activity of eIF-2α. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ APT1 Inhibitor II, Cpd21
A cell permeable acetylpiperazine derivative compound that acts as a selective and reversible inhibitor of lysophospholipase 1 (LYPLA1; IC50 = 840 nM, Ki = 300nM) without affecting the activity of LYPLA2 and 25 other serine hydrolases in mouse BW5147 T cell hydridoma pr
MilliporeSigma™ Calbiochem™ IRE1 Inhibitor IV, KIRA6
KIRA6, IRE1a Kinase Inhibitor.
MilliporeSigma™ Calbiochem™ Bisindolylmaleimide IV
A potent, cell permeable, and selective inhibitor of protein kinase C (IC50 = 87 nM).
MilliporeSigma™ Calbiochem™ Dihydroorotate Dehydrogenase Inhibitor, Brequinar
An immunosuppressive and anti-neoplastic agent that inhibits pyrimidine synthesis by blocking the activity of mammalian mitochondrial dihydroorotate dehydrogenase (DHODH; IC50 = 12 nM).
MilliporeSigma™ Calbiochem™ AMPK Inhibitor, Compound C
AMPK Inhibitor, Compound C, CAS 866405-64-3, is a cell-permeable compound that inhibits KDR/VEGFR2, ALK2/BMPR-I, and AMPK kinase activities (IC50 = 25.1, 148, and 234.6 nM, respectively).
MilliporeSigma™ Calbiochem™ NFAT Inhibitor, MCV1
The NFAT Inhibitor, MCV1 controls the biological activity of NFAT.
MilliporeSigma™ Calbiochem™ TLR8 Agonist, cpd14b
A potent agonist of Toll-like receptor 8 agonist (TLR8, EC50 = 200 nM).
MilliporeSigma™ Calbiochem™ Loperamide Hydrochloride
A very potent and highly selective peripheral resctrictedμ-opioid receptor agonist (Ki = 2
MilliporeSigma™ Calbiochem™ Dipeptidylpeptidase IV Inhibitor I
The Dipeptidylpeptidase IV Inhibitor I controls the biological activity of Dipeptidylpeptidase IV. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ PI 3-Kγ/CKII Inhibitor
The PI 3-Kγ/CKII Inhibitor, also referenced under CAS 1138220-19-5, controls the biological activity of PI 3-Kγ/CKII. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Calpain Inhibitor VI
The Calpain Inhibitor VI, also referenced under CAS 190274-53-4, controls the biological activity of Calpain. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.