SNIPER(BRD)-1 is a SNIPER degrader of BRD4, cIAP1, and XIAP. It has IC50 values of 6.8 nM, 17 nM, and 49 nM for cIAP1, cIAP2, and XIAP, respectively. It can be used for cancer research.
- SNIPER degrader of BRD4, cIAP1, and XIAP.
- IC50 values: cIAP1: 6.8 nM, cIAP2: 17 nM, XIAP: 49 nM.
- Can be used for cancer research.
- Significantly reduces protein levels of BRD4, cIAP1, and XIAP in LNCaP cells.
- Purity: 99.68%.
- Appearance: solid, off-white to light yellow.