Pyrazines
TARGETMOL CHEMICALS INC MIQUELIANIN 10MG
Also available in 5 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Miquelianin (Quercetin 3-glucuronide) is a potent stilbene oxidase inhibitor it has antioxidant anti-atherogenic and anti-inflammatory activities. purity: 98%
TARGETMOL CHEMICALS INC CYANIDIN CHLORIDE 10MG
Also available in 1 mg 5 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Cyanidin Chloride the main phenolic antioxidant in the grape (Vitis vinifera) in particular in the liposomal forms could be used for treatment of diabetes mellitus complications. purity: 98%
TARGETMOL CHEMICALS INC DIHEXA 5MG
Also available in 1 mg 2 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Dihexa (Hexanoyl-Tyr-Ile-Ahx-NH2) is an activator of the hepatocyte growth factor/c-Met (HGF/c-Met) systemit binds to HGF (Kd = 65 pM)and an analog of the peptide angiotensin IV. purity: 98%
TARGETMOL CHEMICALS INC FONDAPARINUX SODIUM 10MG
Also available in 1 mg 2 mg 5 mg 25 mg 50 mg 100 mg and bulk. Please contact Fisher for quotes. Fondaparinux sodium (SR-90107A) is an antithrombin-dependent factor Xa inhibitor with antithrombotic activity. purity: 98%
TARGETMOL CHEMICALS INC DAPANSUTRILE 25MG
Also available in 5 mg 10 mg 50 mg 100 mg 200 mg 500 mg 1000 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Dapansutrile is a potent selective and orally active NLRP3 inflammasome inhibitor with Anti-inflammatory and analgesic activity. purity: 98%
TARGETMOL CHEMICALS INC COLCEMID 10MG
Also available in 1 mg 5 mg 25 mg 50 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Colcemid (NSC-3096) is an inhibitor of microtubule polymerization. It used to study embryonic cloning. purity: 99%
TARGETMOL CHEMICALS INC SCR7 PYRAZINE 10MG
Also available in 1 mg 2 mg 5 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. SCR7 pyrazine (SCR7) enhances CRISPR-Cas9-mediated homology-directed repair (HDR) efficiency in vitro up to 19-fold. Inhibits nonhomologous end-joining (NHEJ). purity: 99%
TARGETMOL CHEMICALS INC NVP-2 5MG
Also available in 1 mg 2 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. NVP-2 is an effective and selective ATP-competitive cyclin-dependent kinase 9 (CDK9) probe. NVP-2 induces cell apoptosis. NVP-2 inhibits CDK9/CycT activity (IC50 0.514 nM). NVP-2 shows inhibitory effcts on CDK1/CycB CDK2/CycA and CDK16/CycY kinases (IC50 0.584 uM 0.706 uM and 0.605 uM respectively). purity: 99%
TARGETMOL CHEMICALS INC PZM21 10MG
Also available in 1 mg 5 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. PZM21 is an effective and selective u opioid receptor agonist (EC50 1.8 nM). purity: 99%
TARGETMOL CHEMICALS INC SR9009 25MG
Also available in 1 mg 2 mg 5 mg 10 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. SR9009 (Stenabolic) a REV-ERB agonist increases the constitutive repression of genes regulated by REV-ERB(alpha)/ERB(beta) (IC50 670/800 nM). Through activation of REV-ERB SR9009 can decrease circadian locomotor activity during the dark phase and alter the expression pattern of core clock genes in the hypothalami of mice. The circadian pattern of expression of an array of metabolic genes in the liver skeletal muscle and adipose tissue was also altered in mice exposed to SR9009 resulting in increased energy expenditure. In Diet-induced obese mice SR9009 (100 mg/kg i.p. b.i.d. for 30 days) could decrease fat mass and markedly improve dyslipidemia and hyperglycemia. purity: 99%
TARGETMOL CHEMICALS INC TELAPREVIR 10MG
Also available in 1 mg 5 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Telaprevir (Incivek) (VX-950) is an effective inhibitor of HCV NS3-4A serine protease (IC50 0.35 uM). purity: 96%
TARGETMOL CHEMICALS INC ML385 25MG
Also available in 5 mg 10 mg 50 mg 100 mg 200 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. ML385 is a new-type and selective NRF2 inhibitor. purity: 99%
TARGETMOL CHEMICALS INC TEPRENONE 500MG
Also available in 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Teprenone (Geranylgeranylacetone) is a anti-ulcer drug and works as an inducer of heat shock proteins (HSPs). purity: 99%
TARGETMOL CHEMICALS INC GEDUNIN 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Gedunin is an important limonoid present in several genera of the Meliaceae family mainly in seeds. Gedunin is an Hsp90 inhibitor and inhibits ovarian cancer cell proliferation. purity: 99%
TARGETMOL CHEMICALS INC YKL-5-124 5MG
Also available in 1 mg 2 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. YKL-5-124 a potent selective and covalent CDK7 inhibitor with an IC50 of 9.7 nM 1300 nM and 3020 nM for CDK7/Mat1/CycH CDK2 and CDK9 respectively displays biochemical and cellular selectivity for CDK7 over CDK12/13. purity: 99%