GSK 1562590 hydrochloride is a high-affinity and selective antagonist of the urotensin-II receptor (UT), with pKis ranging from 9.14 to 9.66 for mammalian recombinant (mouse, rat, cat, monkey, human) and native UT. It is intended for research use only.
- High affinity and selective antagonist of urotensin-II receptor (UT).
- PKis of 9.14-9.66 for mammalian recombinant (mouse, rat, cat, monkey, human) and native UT.
- Appears as a solid, white to off-white in color.
- Soluble in DMSO (25 mg/mL).
- Storage recommendations: -20°C, protect from light, stored under nitrogen; in solvent: -80°C for 6 months; -20°C for 1 month.