Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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2,476
Tocris Bioscience™ GABA
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CAS: 56-12-2 Molecular Formula: C4H9NO2
| CAS | 56-12-2 |
|---|---|
| Molecular Formula | C4H9NO2 |
2,477
Tocris Bioscience™ BX 795
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CAS: 702675-74-9 Molecular Formula: C23H26IN7O2S
| CAS | 702675-74-9 |
|---|---|
| Molecular Formula | C23H26IN7O2S |
2,478
Tocris Bioscience™ LDN 193188
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Inhibitor of phosphatidylcholine transfer protein (PC-TP)
| Target | Lipid Metabolism Inhibitors |
|---|---|
| CAS | 1267610-30-9 |
| Purity | >99% |
| Chemical Name or Material | 2,4-Dichloro-N-[[[4-[[(4,6-dimethyl-2-pyrimidinyl)amino]sulfonyl]phenyl]amino]carbonyl]benzamide |
| Recommended Storage | Store at Room Temperature |
| Molecular Formula | C20H17Cl2N5O4S |
| Formula Weight | 494.35 |
2,479
Tocris Bioscience™ Ipsapirone
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CAS: 95847-70-4 Molecular Formula: C19H23N5O3S
| CAS | 95847-70-4 |
|---|---|
| Molecular Formula | C19H23N5O3S |
2,480
Tocris Bioscience™ DL-Dithiothreitol
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CAS: 12-3-3483 Molecular Formula: C4H10O2S2
| CAS | 12-3-3483 |
|---|---|
| Molecular Formula | C4H10O2S2 |
2,481
Tocris Bioscience™ CGP 36216 hydrochloride
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GABAB antagonist; displays activity at presynaptic receptors
| Inhibitors | CGP 36216 hydrochloride |
|---|---|
| CAS | 1781834-71-6 |
| Product Type | CGP 36216 hydrochloride |
| Molecular Weight (g/mol) | 187.6 |
| Purity | >99% |
2,482
Tocris Bioscience™ CID 16020046
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Selective GPR55 antagonist
| CAS | 834903-43-4 |
|---|---|
| Chemical Name or Material | 4-[4,6-Dihydro-4-(3-hydroxyphenyl)-3-(4-methylphenyl)-6-oxopyrrolo[3,4-c]pyrazol-5(1H)-yl]benzoic acid |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C25H19N3O4 |
| Formula Weight | Observed MW: 425.44 |
| Assay Percent Range | >99% |
2,483
Tocris Bioscience™ CRT 0066854 hydrochloride
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PKCι and PKCζ inhibitor
| Target | Protein Kinase C Inhibitors |
|---|---|
| CAS | 2250019-91-9 |
| Purity | 98% |
| Chemical Name or Material | (2 S)-3-Phenyl-N1-[5,6,7,8-tetrahydro-2-(4-pyridinyl)[1 ]benzothieno[2,3-d]pyrimidin-4-yl]-1,2-propanediamine dihydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C24H25N5S0.2 HCl |
| Formula Weight | Observed MW: 488.48 |
| Assay Percent Range | >98% |
2,484
Tocris Bioscience™ Proglumide sodium salt
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CAS: 99247-33-3 Molecular Formula: C18H25N2NaO4
| CAS | 99247-33-3 |
|---|---|
| Molecular Formula | C18H25N2NaO4 |
2,485
Tocris Bioscience™ WZB 117
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GLUT inhibitor
| CAS | 1223397-11-2 |
|---|---|
| Chemical Name or Material | 3-Fluoro-1,2-phenylene bis(3-hydroxybenzoate) |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C20H13FO6 |
| Formula Weight | Observed MW: 368.31 |
| Assay Percent Range | >98% |
2,486
Tocris Bioscience™ Chroman 1
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Highly potent and selective ROCK 2 inhibitor; improves cell survival after cryogeneisis
| Target | Rho-kinase Inhibitors |
|---|---|
| Purity | 98% |
| Chemical Name or Material | (3 S)-N-[2-[2-(Dimethylamino)ethoxy]-4-(1 H-pyrazol-4-yl)phenyl]-3,4-dihydro-6-methoxy-2 H-1-benzopyran-3-carboxamide dihydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C24H28N4O40.2 HCl |
2,487
Tocris Bioscience™ NPS 2390
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CAS: 226878-01-9 Molecular Formula: C19H21N3O
| CAS | 226878-01-9 |
|---|---|
| Molecular Formula | C19H21N3O |
2,488
Tocris Bioscience™ CCCP
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CAS: 555-60-2 Molecular Formula: C9H5ClN4
| CAS | 555-60-2 |
|---|---|
| Molecular Formula | C9H5ClN4 |
2,489
Tocris Bioscience™ Aliskiren hemifumarate
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Potent renin inhibitor; antihypertensive
| Product Type | Aliskiren hemifumarate |
|---|---|
| Molecular Weight (g/mol) | 609.83 |
| Purity | >99% |
2,490
Tocris Bioscience™ Cycloheximide
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CAS: 66-81-9 Molecular Formula: C15H23NO4
| CAS | 66-81-9 |
|---|---|
| Molecular Formula | C15H23NO4 |