Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Leupeptin, Hemisulfate, Synthetic
Synthetic version of the microbial-derived inhibitor Leupeptin against trypsin-like and cysteine protease activities.
MilliporeSigma™ Calbiochem™ IKKε/TBK1 Inhibitor II, MRT67307
A cell-permeable, potent, ATP-competitive, and reversible dual kinase inhibitor of TBK1/IKKε (IC50 = 19 and 160 nM, respectively).
MilliporeSigma™ Calbiochem™ Cathepsin L Inhibitor III
The Cathepsin L Inhibitor III controls the biological activity of Cathepsin L. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ RuBi-Nicotine
A highly water soluble Ruthenium-bisbipyridine-caged nicotine that can be un-caged by blue and green light
MilliporeSigma™ Calbiochem™ InSolution™ Caspase Inhibitor I
The InSolution™ Caspase Inhibitor I controls the biological activity of Caspase. This small molecule/inhibitor is primarily used for Cancer applications.
MilliporeSigma™ Calbiochem™ CFTR Potentiator, VX-770
A cell-permeable, potentiator of CFTR that directly, reversibly, and allosterically binds to WT and G551D mutant forms (≈10 μM) and increases the open probability to restore lung function.
MilliporeSigma™ Calbiochem™ L3MBTL1 Ligand, UNC669
A nicotinamido-pyrrolidine compound that targets the second MBT (Malignant Brain Tumor) module of chromatin lock L3MBTL1.
MP Biomedicals™ Protease Inhibitor Cocktail Kit
Research Use Only
MilliporeSigma™ Calbiochem™ TMEM16A Activator, Eact
The TMEM16A Activator, Eact modulates the biological activity of TMEM16A. This small molecule/inhibitor is primarily used for Activators/Inducers applications.
MilliporeSigma™ Calbiochem™ Andrographolide
A bicyclic diterpenoid lactone that displays anti-viral, anti-inflammatory, anti-apoptotic, and anti-hyperglycemic properties.
MilliporeSigma™ Calbiochem™ InSolution™ Rho Kinase Inhibitor
The InSolution™ Rho Kinase Inhibitor controls the biological activity of Rho Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ MMP-14 Substrate I, Fluorogenic
A specific fluorescence resonance energy transfer (FRET) peptide substrate for the detection of MMP activity.
MilliporeSigma™ Calbiochem™ β-Amyloid Oligomer Inhibitor, K01-162
The β-Amyloid Oligomer Inhibitor, K01-162 controls the biological activity of β-Amyloid Oligomer.
MilliporeSigma™ Calbiochem™ InSolution™ AG 1478
Highly potent and specific inhibitor of the epidermal growth factor (EGF) receptor tyrosine kinase (IC50 = 3nM)
MilliporeSigma™ Calbiochem™ MTEP Hydrochloride
A non-competitive, potent antagonist highly selective for mGlu5 receptors (IC50 =