Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ TGR5 Receptor Agonist, Cpd23g
A cell-permeable, orally available, phenoxypyrimidine carboxamide derivative that acts as a highly potent and selective agonist of Protein coupled receptor TGR5 (EC50 = 720 pM an
MilliporeSigma™ Calbiochem™ Akt Inhibitor XII, Isozyme-Selective, Akti-2
The Akt Inhibitor XII, Isozyme-Selective, Akti-2 controls the biological activity of Akt. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ PI 3-K/mTOR Inhibitor III, PKI-179
The PI 3-K/mTOR Inhibitor III, PKI-179, also referenced under CAS 1197160-28-3, controls the biological activity of PI 3-K/mTOR. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Ro-32-0432
A selective cell-permeable protein kinase C inhibitor.
MilliporeSigma™ Calbiochem™ p38 MAP Kinase Inhibitor IV
The p38 MAP Kinase Inhibitor IV, also referenced under CAS 1638-41-1, controls the biological activity of p38 MAP Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ IL-2Rα Antagonist
The IL-2Rα Antagonist, also referenced under CAS 1217448-66-2, controls the biological activity of IL-2Rα.
MilliporeSigma™ Calbiochem™ Caspase Modulator II, 1541B
Caspase Modulator II, 1541B primarily used in Inhibition.
MilliporeSigma™ Calbiochem™ Pro-survival Compound, DDD00033325
A cell-permeable, pyrrolidine small molecule that promotes single human embryonic stem cell survival up to 20-fold over background with equal or higher potency than Y-27632.
MilliporeSigma™ Calbiochem™ CRAC Channel Inhibitor, BTP2
The CRAC Channel Inhibitor, BTP2, also referenced under CAS 223499-30-7, controls the biological activity of CRAC Channel. This small molecule/inhibitor is primarily used for Inflammation/Immunology applications.
MilliporeSigma™ Calbiochem™ PP1 Analog V, 2,3-DMB-PP1
A cell-permeable 3-MB-PP1 analog that is more effective than 3-MB-PP1 in inhibiting Syk
MilliporeSigma™ Calbiochem™ Mevastatin, Sodium Salt
Carboxylate form of Mevastatin that is active in whole cells and in cell-free assays.
MilliporeSigma™ Calbiochem™ OSC Inhibitor, Ro 48-8071
The OSC Inhibitor, Ro 48-8071, also referenced under CAS 189197-69-1, controls the biological activity of 2,3-oxidosqualene:lanosterol cyclase activity (OSC).
MilliporeSigma™ Calbiochem™ PP2A Activating Ligand, ITH12246
A cell-permeable, relatively non-toxic, 1,8-naphthyridine derived compound that blocks the inhibitory effect of protein phosphatase inhibitors, such as okadaic acid, on protein phosphatase 2A (PP2A)
MilliporeSigma™ Calbiochem™ REV-ERBα Antagonist, SR8278
The REV-ERBα Antagonist, SR8278 controls the biological activity of REV-ERBα.
MilliporeSigma™ Calbiochem™ 2,3 cis-Piperidine dicarboxylic acid
A non-specific antagonist of NMDA, AMPA and kainate ionotropic receptors and a partial agonist for NMDA receptors.