Lipids and Lipid Derivatives
Medchemexpress LLC Estradiol cypionate | 313-06-4 | MFCD00056558 | 99.5% | 1 ML
Estradiol cypionate is the 17β-cypionate ester of Estradiol, inhibiting ET-1 synthesis by acting on estrogen receptors. It is intended for research use only. In vitro, it inhibits proliferation of gastric cancer cells and induces G1/S phase cell cycle arrest and apoptosis by affecting the PI3K/Akt/mTOR pathway. In vivo, it increases cortical bone density in ovariectomized rabbits, increases occurrence of estrus and pregnancy in cows, and inhibits tumor growth in MGC803 nude mice tumor models.
- Inhibits gastric cancer cell proliferation
- Induces G1/S phase cell cycle arrest and apoptosis
- Increases cortical bone density
- Promotes estrus and pregnancy
- Inhibits tumor growth
Cayman Chemical 2-bromo 17-EstradIol 25mg
A synthetic steroid and inhibitor of estrogen 2-hydroxylase; inhibits estrogen 2-hydroxylase in rat liver microsomes at 50 and 100 µM; prevents estrogen-induced inhibition of apomorphine-induced climbing behavior in mice at 5 mg/kg
Medchemexpress LLC Estra-1,3,5(10)-triene-3,17-diol (17β)-, 3-sulfamate | 172377-52-5 | MFCD00947822 | 351.46 | 25 MG
Estradiol 3-sulfamate, also identified as BLE 00084, E2MATE, or ES-J 995, is characterized as a potent, long-acting, and orally active inhibitor of steroid sulfatase.
- Potent steroid sulfatase inhibitor
- Long-acting steroid sulfatase inhibitor
- Orally active steroid sulfatase inhibitor
- Inhibits estrone sulfatase with an IC50 of 251 nM
- Inhibits estrone sulfatase with a Ki of 133 nM
Selleck Chemical LLC Alpha-Estradiol
Alpha-Estradiol ( -Estradiol 17 alpha-Estradiol Alfatradiol Epiestradiol Epiestrol Alora 17 -E2) a natural non-feminizing stereoisomer a hormonally almost inactive isomer of physiological 17 beta-estradiol (17 -E2) is a weak inhibitor of estrogen
Apexbio Technology LLC Ethinyl Estradiol 57-63-6 100mg
Ethinyl Estradiol (57-63-6) is a small-molecule estrogen receptor agonist targeting intracellular estrogen receptors It is designed to activate these receptors thereby regulating transcription of estrogen-responsive genes and influencing reproductive biology and cell proliferation pathways Ethinyl Estradiol exerts its biological activity primarily through direct binding to estrogen receptors leading to the modulation of endocrine-regulated mechanisms Based on these pharmacological properties Ethinyl Estradiol holds research potential in studies of receptor-mediated responses endocrine regulation mechanisms synthetic hormone interactions drug interactions contraceptive mechanisms and hormone-dependent physiological processes
Sigma Aldrich Fine Chemicals Biosciences Cyproterone acetate European Pharmacopoeia (EP) Reference Standard | 427-51-0 | MFCD00864671 |
Cyproterone acetate European Pharmacopoeia (EP) Reference Standard | Mol Wt: 416.94 | 427-51-0 | MFCD00864671 |
eMolecules 427-51-0 | Medchem Express | Cyproterone acetate | 250mg | 446263199 | HY-13604 | 402.92 | C23H27ClO4
ChemScene | (R)--Methylbenzenepropanamine | 100mg | 726024285 | CS-0029877 | 937-52-0 | MFCD00145208 | 149.237 | C10H15N
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Medchemexpress LLC Estrone-13C3 | 1241684-29-6 | 98.0% | 1 MG
Estrone-13C3 is the 13C-labeled version of Estrone, a naturally occurring estrogenic hormone. It is a primary endogenous estrogen, synthesized in various tissues through the aromatization of androstenedione. This compound is suitable for research use as a tracer and as an internal standard for quantitative analysis.
- Can be used as a tracer
- Can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS
Apexbio Technology LLC Estrone sulfate potassium 1240-04-6 10mg
Estrone sulfate potassium (1240-04-6) is a small-molecule modulator targeting kinase activities implicated in estrogen signaling pathways It is designed to regulate estrogen-mediated biological processes by modulating specific kinase activities thereby influencing cellular responses related to steroid signaling Estrone sulfate potassium exerts its biological activity primarily through modulation of kinase pathways associated with estrogen signaling Laboratory studies indicate that estrone sulfate potassium can influence cellular responses via targeted kinase inhibition pathways Based on these pharmacological properties estrone sulfate potassium holds research potential in elucidating pathological mechanisms and identifying therapeutic targets related to endocrine disorders
Medchemexpress LLC Estradiol 3-methyl ether | 1035-77-4 | 99.9% | 286.41 | 25 MG
Estradiol 3-methyl ether is a synthetic estrogen. It can disrupt microtubule networks in V79 cells with an EC50 of 9 μM and inhibits cell proliferation. Estradiol 3-methyl ether has also been shown to decrease serum cholesterol levels and increase body weight loss, indicating feminizing activity in an HFD murine model.
- Synthetic estrogen
- Disrupts microtubule networks in V79 cells (EC50 of 9 μM)
- Inhibits cell proliferation
- Decreases serum cholesterol levels
- Increases body weight loss in HFD murine models
Medchemexpress LLC Estradiol 3-sulfamate | 172377-52-5 | 351.46 | 50 MG
Estradiol 3-sulfamate is a potent, long-acting, and orally active steroid sulfatase inhibitor. It inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. The compound is readily transformed and absorbed in the gut into its oxidative metabolite, EMATE, demonstrating potent and long-acting STS inhibition.
- Potent, long-acting, and orally active steroid sulfatase inhibitor.
- Inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM.
- Increased estrone sulfatase inhibitory activity with specific halogen moieties.
- Readily absorbed and transformed in the gut into its oxidative metabolite, EMATE.
- Both compounds demonstrate potent and long-acting STS inhibition.
Apexbio Technology LLC Ethinyl Estradiol 57-63-6 500mg
Ethinyl Estradiol (57-63-6) is a small-molecule estrogen receptor agonist targeting intracellular estrogen receptors It is designed to activate these receptors thereby regulating transcription of estrogen-responsive genes and influencing reproductive biology and cell proliferation pathways Ethinyl Estradiol exerts its biological activity primarily through direct binding to estrogen receptors leading to the modulation of endocrine-regulated mechanisms Based on these pharmacological properties Ethinyl Estradiol holds research potential in studies of receptor-mediated responses endocrine regulation mechanisms synthetic hormone interactions drug interactions contraceptive mechanisms and hormone-dependent physiological processes
Cayman Chemical 2-bromo 17-EstradIol 50mg
A synthetic steroid and inhibitor of estrogen 2-hydroxylase; inhibits estrogen 2-hydroxylase in rat liver microsomes at 50 and 100 µM; prevents estrogen-induced inhibition of apomorphine-induced climbing behavior in mice at 5 mg/kg
Innovative Reseach Of America INNOVATIVE RESEARCH OF AMERICA
NC3903870 0.36 MG 17B ESTRADIOL PELLETS