(Rac)-5-Hydroxymethyl Tolterodine, also known as (Rac)-Desfesoterodine, is an active metabolite of Tolterodine. It acts as a mAChR antagonist, targeting M1-M5 receptors with specific Ki values ranging from 2.3 nM to 2.9 nM. This compound is primarily utilized in research related to overactive bladder. It presents as a solid, white to off-white substance.
- Functions as a mAChR antagonist
- Targets M1, M2, M3, M4, and M5 receptors
- Used for overactive bladder research
- Solid, white to off-white appearance
- Molecular weight of 341.50
- Inhibits carbachol-induced contraction in guinea-pig urinary bladder strips
- Exhibits significant muscarinic receptor binding activity