Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ MAP Kinase Inhibitor Set I
The MAP Kinase Inhibitor Set I controls the biological activity of MAP Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Adenosine 3',5'-cyclic Monophosphate, N6-Benzoyl-, Sodium Salt
A potent cell-permeable activator of cAMP-dependent protein kinase (PKA).
MilliporeSigma™ Calbiochem™ Insulin Expression Inducer, BRD7389
A cell-permeable naphthoquinolinedione compound that specifically induces insulin secretion in mouse αTC1-cells and promotes transdifferentiation to a β-cell-like status.
MilliporeSigma™ Calbiochem™ Tiagabine Hydrochloride
A potent uptake inhibitor highly selective for GABA Transport-1 (IC50 = 67nM in vivo
MilliporeSigma™ Calbiochem™ CTAP
A highly potent octapeptide that acts as a selective and brain penetrating bioavailableμ opioid receptor antagonist (IC50
MilliporeSigma™ Calbiochem™ TACE Substrate IV, Fluorogenic
An internally-quenched fluorogenic decapeptide substrate that is useful for continuous monitoring of TACE activity and high-throughput screening of TACE inhibitors (kcat =
MilliporeSigma™ Calbiochem™ PDE4D Inhibitor, GEBR-7b
The PDE4D Inhibitor, GEBR-7b controls the biological activity of PDE4D. This small molecule/inhibitor is primarily used for Cell Signaling applications.
MilliporeSigma™ Calbiochem™ Interleukin-1 Receptor-Associated-Kinase-1/4 Inhibitor
The Interleukin-1 Receptor-Associated-Kinase-1/4 Inhibitor controls the activity of Interleukin-1 Receptor-Associated-Kinase-1/4. Primarily used for Phosphorylation & Dephosphorylation apps.
MilliporeSigma™ Calbiochem™ Plasminogen Activator Inhibitor-1, Human, Recombinant
Primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ Polo-like Kinase Inhibitor II, BTO-1
The Polo-like Kinase Inhibitor II, BTO-1, also referenced under CAS 40647-02-7, controls the biological activity of Polo-like Kinase. This small molecule/inhibitor is primarily used for Phosphorylation and Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ SKP2 E3 Ligase Inhibitor IV
A cell-permeable inhibitor of SKP2-dependent p27Kip1 ubiquitination. Selectively induces the accumulation SCFSKP2 substrates in multiple myeloma RPMI 8226 cells.
MilliporeSigma™ Calbiochem™ REV-ERBα Agonist, GSK4112
The REV-ERBα Agonist, GSK4112 controls the biological activity of REV-ERBα. This small molecule/inhibitor is primarily used for Biochemicals applications.
MilliporeSigma™ Calbiochem™ ETV1 Inhibitor, BRD32048
Cell-permeable, reversibly binds to ETV1 (KD = 17.1 μM) and reduces its transcriptional activity, independent of its binding to DNA.
MilliporeSigma™ Calbiochem™ PI 3-Kα Inhibitor IV
The PI 3-Kα Inhibitor IV, also referenced under CAS 1188890-32-5, controls the biological activity of PI 3-Kα. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Lactate Dehydrogenase A Inhibitor, FX11
Lactate Dehydrogenase A Inhibitor, FX11, CAS 213971-34-7, is a cell permeable, selective, reversible, NADH competitive inhibitor of lactate dehhydrogenase A (LDHA; Ki = 8μM for human liver LDHA).