Lipids and Lipid Derivatives
Medchemexpress LLC CGGK acetate | 96.78% | 363.43 (free acid) | 1 MG
CGGK acetate is a control peptide of CAQK peptide, intended for research use only. It presents as a white to off-white solid with a purity of 96.78% and a molecular weight of 363.43 (free acid). Its chemical formula is C13H25N5O5S.xC2H4O2. This product is shipped at room temperature and requires sealed storage, away from moisture.
- Sequence: Cys-Gly-Gly-Lys
- Purity: 96.78%
- Solubility in DMSO: ≥ 100 mg/mL
- Powder storage: -80°C for 2 years, or -20°C for 1 year
- In solvent storage: -80°C for 6 months, or -20°C for 1 month
Medchemexpress LLC AKN-028 acetate | 98.4% | 362.39 | 50 MG
AKN-028 acetate is a novel tyrosine kinase (TK) inhibitor. It is a potent, orally active FMS-like receptor tyrosine kinase 3 (FLT3) inhibitor with an IC50 value of 6 nM. It inhibits FLT3 autophosphorylation and induces a dose-dependent cytotoxic response (mean IC50=1 μM). It also induces apoptosis by activation of caspase 3. AKN-028 acetate can be used in research of acute myeloid leukemia (AML).
- Novel tyrosine kinase (TK) inhibitor
- Potent, orally active FMS-like receptor tyrosine kinase 3 (FLT3) inhibitor with an IC50 value of 6 nM
- Inhibits FLT3 autophosphorylation
- Induces a dose-dependent cytotoxic response (mean IC50=1 μM)
- Induces apoptosis by activation of caspase 3
- Can be used in research of acute myeloid leukemia (AML)
- Inhibits growth of primary AML and MV4-11 cells in mice
Medchemexpress LLC Megestrol acetate (Standard) | 595-33-5 | 98.5% | 384.51 | 50 MG
Megestrol acetate (Standard) is the analytical standard of Megestrol acetate, intended for research and analytical applications. It is a synthetic and orally active progesteronal agent. This product is effective as an appetite stimulant for wasting syndromes like cachexia and decreases nuclear and cytosol androgen receptors in human BPH tissue. It also has potential for HIV study and downregulates the autophagic catabolic pathway.
- Effective as an appetite stimulant for wasting syndromes
- Decreases nuclear and cytosol androgen receptors in human BPH tissue
- Potential for HIV study
- Downregulates the autophagic catabolic pathway
- Suitable for qualitative, quantitative, and methodological research in HPLC, GC, and MS
Medchemexpress LLC Retinyl acetate | 127-47-9 | 328.49 | 1 ML
Retinyl acetate is a synthetic acetate ester form derived from retinol that possesses potential antineoplastic and chemopreventive activities. It is for research use only and not sold to patients.
- Purity of 99.30%
- Off-white to light yellow solid appearance
- Classified as terpenoids, diterpenoids
- Initial source is endogenous metabolite
- Shipped at room temperature in continental US
- Store powder at -20°C for 3 years
- Store in solvent at -80°C for 6 months or -20°C for 1 month
- Inhibits proliferation of tumor cells at 10 μM in vitro
- Inhibits DMBA induced mammary carcinogenesis in Sprague-Dawley rats at 250 mg/kg in diet in vivo
Apexbio Technology LLC Guanabenz Acetate 23256-50-0 50mg
Guanabenz Acetate (CAS 23256-50-0) is a small molecule that acts as a selective agonist of the 2-adrenergic receptor subtypes It exhibits notable affinity for the 2a-adrenergic receptor (pEC50 8 25) with moderate activity at the 2b-adrenergic receptor (pEC50 7 01) and lower potency at the 2c-adrenergic receptor (pEC50 5) Through activation of these receptors Guanabenz Acetate modulates adrenergic neurotransmission making it a valuable tool for investigating the physiological and pharmacological functions of 2-adrenergic signaling in biomedical research
Medchemexpress LLC Poneratoxin acetate | 2756.35 (free base) | 10 MG
Poneratoxin acetate is the acetate salt form of Poneratoxin (HY-P10234). It acts as a modulator for voltage-gated sodium channels (NaV, with EC50 for NaV1.6 and NaV1.7 being 97 nM and 2.3 μM), decreasing the voltage threshold for activation and inhibiting channel inactivation. This compound enhances the excitability of neurons and contributes to the transmission of pain signals.
- Modulator for voltage-gated sodium channels
- Lowers the voltage threshold for activation
- Inhibits the inactivation of channels
- Enhances the excitability of neurons
- Contributes to the transmission of pain signals
- For powder, store at -80°C for 2 years or -20°C for 1 year
- For solution, store at -80°C for 6 months or -20°C for 1 month
- Store sealed and away from moisture
Medchemexpress LLC CBP-501 (acetate) | 1929.06 (free base) | 1 MG
CBP-501 acetate is a cell-permeable calmodulin-binding peptide and a G2-abrogating drug candidate. It inhibits the activity of multiple Ser216-specific kinases, including MAPKAP-K2, C-Tak1, CHK1, and CHK2. It is used for various types of cancer and enhances the cytotoxicity of CDDP and Bleomycin against cancer cells both in vitro and in vivo.
- Inhibits MAPKAP-K2 with an IC50 of 0.9 μM
- Inhibits C-Tak1 with an IC50 of 1.4 μM
- Inhibits Chk1 with an IC50 of 3.4 μM
- Inhibits Chk2 with an IC50 of 6.5 μM
- Stable for 2 years at -80°C as powder
- Stable for 1 year at -20°C as powder
- Stable for 6 months at -80°C in solvent
- Stable for 1 month at -20°C in solvent
- Enhances cytotoxicity of CDDP and Bleomycin
Medchemexpress LLC Farnesyl pyrophosphate ammonium | 116057-57-9 | 95.39% | 433.42 | 1 MG
Farnesyl pyrophosphate ammonium is a metabolic intermediate in the mevalonate (MVA) pathway. It acts as a TRP channel (TRPM2) agonist, triggering Ca2+ influx and cell death. It is a crucial branch substrate for various biological syntheses and is utilized in research concerning a range of diseases.
- Acts as a TRP channel (TRPM2) agonist
- Triggers Ca2+ influx and cell death
- Key branch substrate for cholesterol synthesis
- Key branch substrate for ubiquinone synthesis
- Key branch substrate for protein farnesylation
- Key branch substrate for geranylgeranyl pyrophosphate (GGPP) synthesis
- Used in research on cerebral ischemia
- Used in research on neurodegenerative diseases
- Used in research on pancreatic cancer
- Used in research on inflammation
- Used in research on autoimmune diseases
TARGETMOL CHEMICALS INC OCTREOTIDE ACETATE 100MG
Also available in 5 mg 10 mg 25 mg 50 mg 200 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Octreotide Acetate (Sandostatin) is a potent long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone. purity: 99%
Medchemexpress LLC Goserelin (acetate) | 145781-92-6 | MFCD01747329 | 99.9% | C61H88N18O16 | 10MG
Goserelin (acetate) is a synthetic decapeptide analog of gonadotropin-releasing hormone (GnRH) used as a research-grade GnRH agonist for in vitro and in vivo studies of hormone-dependent cancers, reproductive biology, and endocrine signaling. Provided as the acetate salt with high analytical purity, it is supplied as a white to off-white solid and intended for research use only.
- Purity 99.9% (HPLC).
- Molecular formula C61H88N18O16 and molecular weight 1329.46.
- White to off-white solid suitable for analytical and biological assays.
- Supplied in small vial sizes suitable for dosing and assay development.
- Stable when stored sealed, away from moisture; powder: -80°C (up to 2 years), -20°C (up to 1 year).
- Acetate salt form for standard biochemical handling.
- For research use only; not for human or veterinary use.
Medchemexpress LLC Delmitide acetate 10mg | 501019-16-5 | 10MG
Delmitide (RDP58) acetate is an orally active d-isomer decapeptide with potent anti-inflammatory activity Delmitide acetate inhibits production of TNF- IFN- and interleukin (IL)-12 and up-regulates heme oxygenase 1 activity Delmitide acetate can be used for the research of ulcerative colitis[1 [2
Sigma Aldrich Fine Chemicals Biosciences Octyl beta D glucopyranosi10G
Octyl beta D glucopyranosi10G
Medchemexpress LLC Flecainide acetate | 54143-56-5 | MFCD00214290 | 99.4% | 474.39 g/mol | C19H24F6N2O5 | 10 MG
Flecainide acetate is a class 1C antiarrhythmic research reagent that inhibits cardiac Nav1.5 sodium channels. Supplied as a white to off-white solid for laboratory use; intended for research use only and not for human or clinical use.
- Class 1C antiarrhythmic agent that blocks Nav1.5 sodium channels.
- Supplied as a white to off-white solid suitable for analytical and biological research.
- High purity of 99.4%.
- Molecular formula C19H24F6N2O5; molecular weight 474.39 g/mol.
- Available in small research pack sizes, including 10 mg.
- Store solid at 4°C; store solutions at -80°C (up to 6 months) or -20°C (up to 1 month).
Cayman Chemical DL-Tryptophan octyl ester (hydrochloride), Purity: ≥98%, CAS: 6278-90-6, 5 g
A stable, cell-permeable tryptophan derivative with an octyl ester protected COOH group
Medchemexpress LLC Rezafungin acetate 10mM 1mL | 1631754-41-0 | 10MM 1ML
Rezafungin acetate (Biafungin acetate) is a next-generation broad-spectrum and long-lasting echinocandin Rezafungin acetate shows potent antifungal activity against Candida spp Aspergillus spp and Pneumocystis spp [1 [2